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Theliatinib
Theliatinib is a small molecule pharmaceutical. It is currently being investigated in clinical studies. The pharmaceutical is active against epidermal growth factor receptor. In addition, it is known to target tyrosine-protein kinase Lck, receptor tyrosine-protein kinase erbB-4, tyrosine-protein kinase Yes, non-receptor tyrosine-protein kinase TNK1, and tyrosine-protein kinase Lyn.
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Commercial
Therapeutic Areas
No data
Trade Name
FDA
EMA
No data
Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
No data
Labels
FDA
EMA
No data
Indications
FDA
EMA
No data
Agency Specific
FDA
EMA
No data
Patent Expiration
No data
ATC Codes
No data
HCPCS
No data
Clinical
Clinical Trials
2 clinical trials
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Mock data
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Indications Phases 4
No data
Indications Phases 3
No data
Indications Phases 2
No data
Indications Phases 1
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
NeoplasmsD009369C802————2
Indications Without Phase
No data
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameTHELIATINIB
INNxiliertinib
Description
Theliatinib is a small molecule pharmaceutical. It is currently being investigated in clinical studies. The pharmaceutical is active against epidermal growth factor receptor. In addition, it is known to target tyrosine-protein kinase Lck, receptor tyrosine-protein kinase erbB-4, tyrosine-protein kinase Yes, non-receptor tyrosine-protein kinase TNK1, and tyrosine-protein kinase Lyn.
Classification
Small molecule
Drug classtyrosine kinase inhibitors
Image (chem structure or protein)
Structure (InChI/SMILES or Protein Sequence)—
Identifiers
PDB—
CAS-ID1353644-70-8
RxCUI—
ChEMBL IDCHEMBL3545180
ChEBI ID—
PubChem CID—
DrugBank—
UNII ID6ZZ3B7NZ0B (ChemIDplus, GSRS)
Target
Agency Approved
EGFR
EGFR
Organism
Homo sapiens
Gene name
EGFR
Gene synonyms
ERBB, ERBB1, HER1
NCBI Gene ID
1956
Protein name
epidermal growth factor receptor
Protein synonyms
avian erythroblastic leukemia viral (v-erb-b) oncogene homolog, cell growth inhibiting protein 40, cell proliferation-inducing protein 61, EGFR vIII, epidermal growth factor receptor tyrosine kinase domain, erb-b2 receptor tyrosine kinase 1, Proto-oncogene c-ErbB-1, Receptor tyrosine-protein kinase erbB-1
Uniprot ID
Q9UMG5
Mouse ortholog
Egfr (13649)
epidermal growth factor receptor (Q01279)
Alternate
LCK
LCK
ERBB4
ERBB4
YES1
YES1
TNK1
TNK1
LYN
LYN
Organism
Homo sapiens
Gene name
LCK
Gene synonyms
NCBI Gene ID
3932
Protein name
tyrosine-protein kinase Lck
Protein synonyms
Leukocyte C-terminal Src kinase, LSK, Lymphocyte cell-specific protein-tyrosine kinase, p56(LSTRA) protein-tyrosine kinase, p56-LCK, Protein YT16, Proto-oncogene Lck, proto-oncogene tyrosine-protein kinase LCK, T cell-specific protein-tyrosine kinase, T-lymphocyte specific protein tyrosine kinase p56lck
Uniprot ID
Q9NYT8
Mouse ortholog
Lck (16818)
proto-oncogene tyrosine-protein kinase LCK (Q91X65)
Variants
Clinical Variant
No data
Financial
No data
Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 5 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
0 adverse events reported
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